Journal of Medicinal Chemistry
Volume 39, Issue 4 (February 16, 1996)
Copyright © 1996
American Chemical Society
811-813 | Bis(31/31'){[Cys31,Trp32,Nva34]NPY- (31-36)}: A Specific NPY Y-1 Receptor Antagonist
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814-816 | (2S,4S)-2-Amino-4-(4,4-diphenylbut-1-yl)- pentane-1,5-dioic Acid: A Potent and Selective Antagonist for Metabotropic Glutamate Receptors Negatively Linked to Adenylate Cyclase
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817-825 | Novel 3-Pyridyl Ethers with Subnanomolar Affinity for Central Neuronal Nicotinic Acetylcholine Receptors
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826-833 | In Vivo Biodistribution, Pharmacokinetic Parameters, and Brain Uptake of 5-Halo-6-methoxy(or ethoxy)-5,6-dihydro-3'-azido-3'-deoxythymidine Diastereomers as Potential Prodrugs of 3'-Azido-3'-deoxythymidine
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834-841 | Tetrahydronaphthalenes: Influence of Heterocyclic Substituents on Inhibition of Steroidogenic Enzymes P450 arom and P450 17
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842-849 | Controlled Modification of Acidity in Cholecystokinin B Receptor Antagonists: N-(1,4-Benzodiazepin-3-yl)-N '-[3-(tetrazol-5-ylamino)phenyl]ureas
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850-859 | Comparative Molecular Field Analysis-Based Prediction of Drug Affinities at Recombinant D1A Dopamine Receptors
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860-872 | Synthesis, Biological Evaluation, and Quantitative Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as Novel Tifluadom-like Ligands with High Affinity and Selectivity for -Opioid Receptors
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873-880 | Synthesis of Non-nucleoside Analogs of Toyocamycin, Sangivamycin, and Thiosangivamycin: Influence of Various 7-Substituents on Antiviral Activity
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881-891 | Structure-Activity Relationships among 2-Substituted 5,6-Dichloro-, 4,6-Dichloro-, and 4,5-Dichloro-1-[(2-hydroxyethoxy)methyl]- and -1-[(1,3-dihydroxy-2-propoxy)methyl]benzimidazoles
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892-903 | High-Affinity Inhibitors of Dihydrofolate Reductase: Antimicrobial and Anticancer Activities of 7,8-Dialkyl-1,3-diaminopyrrolo[3,2-f]quinazolines with Small Molecular Size
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904-917 | Structure-Based Design of Lipophilic Quinazoline Inhibitors of Thymidylate Synthase
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918-928 | Tyrosine Kinase Inhibitors. 9. Synthesis and Evaluation of Fused Tricyclic Quinazoline Analogues as ATP Site Inhibitors of the Tyrosine Kinase Activity of the Epidermal Growth Factor Receptor
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929-936 | Highly Selective Bradykinin Agonists and Antagonists with Replacement of Proline Residues by N-Methyl-D- and L-phenylalanine
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937-948 | 3- and 4-Substituted 4H-Pyrido[4,3-e]-1,2,4-thiadiazine 1,1-Dioxides as Potassium Channel Openers: Synthesis, Pharmacological Evaluation, and Structure-Activity Relationships
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949-956 | Guanine, Pyrazolo[3,4-d]pyrimidine, and Triazolo[4,5-d]pyrimidine (8-Azaguanine) Phosphonate Acyclic Derivatives as Inhibitors of Purine Nucleoside Phosphorylase
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957-967 | Azole Endothelin Antagonists. 1. A Receptor Model Explains an Unusual Structure-Activity Profile
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968-981 | Azole Endothelin Antagonists. 2. Structure-Activity Studies
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982-991 | Azole Endothelin Antagonists. 3. Using log P as a Tool To Improve Absorption
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992-998 | Substituted 2,5'-Bi-1H-benzimidazoles: Topoisomerase I Inhibition and Cytotoxicity
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999-1004 | Homologs of Idoxifene: Variation of Estrogen Receptor Binding and Calmodulin Antagonism with Chain Length
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1005-1008 | Selectively Cytotoxic Diterpenes from Euphorbia poisonii
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1009-1009 | Synthesis and Applications of Isotopically Labelled Compounds 1994. Proceedings of the Fifth International Symposium, Strasbourg France, 20-24 June, 1994 Edited by J. Allen and R. Voges. John Wiley & Sons, New York. 1995. xxix + 935 pp. 15.5 × 23.5 cm. ISBN 0-471-95143-9. $199.95.
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1009-1009 | Oxidative Stress, Lipoproteins and Cardiovascular Dysfunction. Portland Press Research Monograph VII Edited by C. Rice-Evans and K. R. Bruckdorfer. Portland Press Ltd., London. 1995. xvi + 184 p. 15.5 × 23.5 cm. ISBN 1-85587-045-3. $96.00.
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1009-1010 | Biochemistry of Redox Reactions By B. Testa. Academic Press, New York. 1995. xviii + 471 pp. 19.4 × 26.2 cm. ISBN 0-12-685391-6. $75.00.
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1010-1010 | The Logic of Chemical Synthesis By E. J. Corey and Xue-Min Cheng. John Wiley & Sons, Inc., New York. 1995. 436 pp. 18 × 25 cm. ISBN 0-471-11594-0. $24.95 (pbk).
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1010-1011 | Fundamentals of Enzyme Kinetics. Revised Edition By Athel Cornish-Bowden. Portland Press, London. 1995. xiii + 343 pp. 17.5 cm × 24.5 cm. ISBN 1-85578-072-0. $29.00.
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1011-1011 | New Perspectives in Drug Design Edited by P. M. Dean, G. Jolles, and C. G. Newton. Academic Press Inc., San Diego, CA. 1995. xiv + 321 pp. 15.5 × 23.5 cm. ISBN 0-12-208070-x. $50.00.
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1011-1011 | Biochemistry of Cell Membranes. A Compendium of Selected Topics Edited by S. Papa and J. M. Tager. Birkhauser Verlag, Basel, Switzerland. 1995. viii + 365 pp. 16 × 24 cm. ISBN 3-7643-5056-3. $149.00.
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1011-1012 | The Golden Helix. Inside Biotech Ventures By Arthur Kornberg. University Science Books, Sausalito, CA. 1995. xi + 287 pp. 16 × 24 cm. ISBN 0-935702-32-6. $28.50.
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1012-1012 | Diazo Chemistry By Heinrich Zollinger. VCH Verlagsgesellschaft mbH, Weinheim, Germany. I. Aromatic and Heteroaromatic Compounds. 1994. xiii + 453 pp. 17.5 × 24.5 cm. ISBN 3-527-29213-6. DM 198.00; II. Aliphatic, Inorganic and Organometallic Compounds. 1995. xvi + 522 pp. 17.5 × 24.5 cm. ISBN 3-527-29222-5. DM 174.00. Set ISBN 3-527-29328-0. DM 348.00.
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