3229-3234
| Identification of the First Retinoid X Receptor Homodimer Antagonist
Stacie S. Canan Koch,
Laura J. Dardashti,
Jonathan J. Hebert,
Steven K. White,
Glenn E. Croston,
Karen S. Flatten,
Richard A. Heyman, and
Alex M. Nadzan
[Full Article -
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3235-3237
| (S)-(-)-5-Ethynyl-3-(1-methyl-2-pyrroli- dinyl)pyridine Maleate (SIB-1508Y): A Novel Anti-Parkinsonian Agent with Selectivity for Neuronal Nicotinic Acetylcholine Receptors
Nicholas D. P. Cosford,
Leo Bleicher,
Audrey Herbaut,
J. Stuart McCallum,
Jean-Michel Vernier,
Heather Dawson,
Jeffrey P. Whitten,
Pamala Adams,
Laura Chavez-Noriega,
Lucia D. Correa,
James H. Crona,
Lorrence S. Mahaffy,
Frederique Menzaghi,
Tadimeti S. Rao,
Richard Reid,
Aida I. Sacaan,
Emily Santori,
Kenneth A. Stauderman,
Kevin Whelan,
G. Kenneth Lloyd, and
Ian A. McDonald
[Full Article -
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3238-3240
| Structural Modifications of Thalidomide Produce Analogs with Enhanced Tumor Necrosis Factor Inhibitory Activity
George W. Muller,
Laura G. Corral,
Mary G. Shire,
Hua Wang,
Andre Moreira,
Gilla Kaplan, and
David I. Stirling
[Full Article -
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3241-3247
| Synthesis and Growth Inhibitory Properties of Glycosides of 1-O-Hexadecyl-2-O-methyl-sn-glycerol, Analogs of the Antitumor Ether Lipid ET-18-OCH3 (Edelfosine)
José R. Marino-Albernas,
Robert Bittman,
Andrew Peters, and
Eric Mayhew
[Full Article -
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3248-3255
| Synthesis and Structure-Activity Relationships of 1,2,3,4-Tetrahydroquinoline-2,3,4-trione 3-Oximes: Novel and Highly Potent Antagonists for NMDA Receptor Glycine Site
Sui Xiong Cai,
Zhang-Lin Zhou,
Jin-Cheng Huang,
Edward R. Whittemore,
Zizi O. Egbuwoku,
Yixin Lü,
Jon E. Hawkinson,
Richard M. Woodward,
Eckard Weber, and
John F. W. Keana
[Full Article -
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3256-3262
| Synthesis and in Vitro and in Vivo Characteristics of an Iodinated Analogue of the  -Adrenoceptor Antagonist Carazolol
Eric A. Dubois,
Jan C. van den Bos,
Tamme Doornbos,
Peter A. P. M. van Doremalen,
G. Aernout Somsen,
Jozef A. J. M. Vekemans,
Anton G. M. Janssen,
Harry D. Batink,
Gerard J. Boer,
Martin Pfaffendorf,
Eric A. van Royen, and
Pieter A. van Zwieten
[Full Article -
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3263-3268
| Synthesis of 2'-Aminomethyl Derivatives of N-(2-(Phosphonomethoxy)ethyl) Nucleotide Analogues as Potential Antiviral Agents
Hana Dvoáková,
Milena Masojídková,
Antonín Hol,
Jan Balzarini,
Graciela Andrei,
Robert Snoeck, and
Erik De Clercq
[Full Article -
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3269-3277
| 3-(2-Benzofuranyl)quinuclidin-2-ene Derivatives: Novel Muscarinic Antagonists
Gunnar Nordvall,
Staffan Sundquist,
Gary Johansson,
Gunilla Glas,
Lisbeth Nilvebrant, and
Uli Hacksell
[Full Article -
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3278-3290
| Nonpeptidal P2 Ligands for HIV Protease Inhibitors: Structure-Based Design, Synthesis, and Biological Evaluation
Arun K. Ghosh,
John F. Kincaid,
D. Eric Walters,
Yan Chen,
Narayan C. Chaudhuri,
Wayne J. Thompson,
Chris Culberson,
Paula M. D. Fitzgerald,
Hee Yoon Lee,
Sean P. McKee,
Peter M. Munson,
Tien T. Duong,
Paul L. Darke,
Joan A. Zugay,
William A. Schleif,
Melinda G. Axel,
Juinn Lin, and
Joel R. Huff
[Full Article -
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3291-3299
| Paracyclophanes: A Novel Class of Water-Soluble Inhibitors of HIV Proteinase
Peter Ettmayer,
Andreas Billich,
Peter Hecht,
Brigitte Rosenwirth, and
Hubert Gstach
[Full Article -
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3300-3306
| Phosphodiester Amidates of Allenic Nucleoside Analogues: Anti-HIV Activity and Possible Mechanism of Action
Holger Winter,
Yosuke Maeda,
Hiroaki Mitsuya, and
Jiri Zemlicka
[Full Article -
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3307-3318
| Synthesis and Antiviral Activity Evaluation of Some New Aminoadamantane Derivatives. 2
Nicolas Kolocouris,
Antonios Kolocouris,
George B. Foscolos,
George Fytas,
Johan Neyts,
Elisabeth Padalko,
Jan Balzarini,
Robert Snoeck,
Graciela Andrei, and
Erik De Clercq
[Full Article -
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3319-3323
| 3- and 4-Pyridylalkyl Adamantanecarboxylates: Inhibitors of Human Cytochrome P45017 (17-Hydroxylase/C17,20-Lyase). Potential Nonsteroidal Agents for the Treatment of Prostatic Cancer
Ferdinand C. Y. Chan,
Gerard A. Potter,
S. Elaine Barrie,
Benjamin P. Haynes,
Martin G. Rowlands,
John Houghton, and
Michael Jarman
[Full Article -
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3324-3330
| A Single-Point Slight Alteration Set as a Tool for Structure-Activity Relationship Studies of Ovine Corticotropin Releasing Factor
Michael Beyermann,
Klaus Fechner,
Jens Furkert,
Eberhard Krause, and
Michael Bienert
[Full Article -
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3331-3342
| Vesamicol Receptor Mapping of Brain Cholinergic Neurons with Radioiodine- Labeled Positional Isomers of Benzovesamicol
Yong-Woon Jung,
Kirk A. Frey,
G. Keith Mulholland,
Renato del Rosario,
Phillip S. Sherman,
David M. Raffel,
Marcian E. Van Dort,
David E. Kuhl,
David L. Gildersleeve, and
Donald M. Wieland
[Full Article -
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3343-3356
| New Low-Density Lipoprotein Receptor Upregulators Acting via a Novel Mechanism
Michael J. Ashton,
Thomas J. Brown,
Garry Fenton,
Frank Halley,
Mark F. Harper,
Peter M. Lockey,
Barry Porter,
Alan G. Roach,
Keith A. J. Stuttle,
Nigel Vicker, and
Roger J. A. Walsh
[Full Article -
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3357-3366
| Mechanistic Studies on the Inactivation of Papain by Epoxysuccinyl Inhibitors
Joseph P. Meara and
Daniel H. Rich
[Full Article -
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3367-3374
| Design, Synthesis, and Biological Evaluation of Ellipticine-Estradiol Conjugates
Rajesh Devraj,
John F. Barrett,
Jeffrey A. Fernandez,
John A. Katzenellenbogen, and
Mark Cushman
[Full Article -
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3375-3384
| Antitumor Benzothiazoles. 3. Synthesis of 2-(4-Aminophenyl)benzothiazoles and Evaluation of Their Activities against Breast Cancer Cell Lines in Vitro and in Vivo
Dong-Fang Shi,
Tracey D. Bradshaw,
Samantha Wrigley,
Carol J. McCall,
Peter Lelieveld,
Iduna Fichtner, and
Malcolm F. G. Stevens
[Full Article -
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3385-3393
| Synthesis and Quantitative Structure-Activity Relationships of 17-(Hydrazonomethyl)-5-androstane-3,14-diol Derivatives That Bind to Na+,K+-ATPase Receptor
Luisa Quadri,
Alberto Cerri,
Patrizia Ferrari,
Elena Folpini,
Massimo Mabilia, and
Piero Melloni
[Full Article -
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3394-3400
| Quantitative Structure-Activity Relationships for the in Vitro Antimycobacterial Activity of Pyrazinoic Acid Esters
Kathryn E. Bergmann,
Michael H. Cynamon, and
John T. Welch
[Full Article -
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3401-3408
| Molecular Similarity Based on DOCK-Generated Fingerprints
Hans Briem and
Irwin D. Kuntz
[Full Article -
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3409-3411
| Antitumor Activity of S-(p-Bromobenzyl)glutathione Diesters in Vitro: A Structure-Activity Study
Paul J. Thornalley,
Muhati J. Ladan,
Simon J. S. Ridgway, and
Yubin Kang
[Full Article -
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3412-3417
| Synthesis and Evaluation of Novel Thymidine Analogs as Antitumor and Antiviral Agents
Xiannong Chen,
Kenneth Bastow,
Barry Goz,
Louis S. Kucera,
Susan L. Morris-Natschke, and
Khalid S. Ishaq
[Full Article -
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3418-3422
| Synthesis and Antiretroviral Evaluation of New Alkoxy and Aryloxy Phosphate Derivatives of 3'-Azido-3'-deoxythymidine
Andrew Tsotinis
, Theodora Calogeropoulou,
Maria Koufaki, and
Charikleia Souli
, Jan Balzarini and
Erik De Clercq
, Alexandros Makriyannis
[Full Article -
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3423-3428
| (±)-3-[4'-(N,N-Dimethylamino)cinnamyl]benzazepine Analogs: Novel Dopamine D1 Receptor Antagonists
Jamshed H. Shah,
Richard H. Kline,
Beth Geter-Douglass,
Sari Izenwasser,
Jeffrey M. Witkin, and
Amy Hauck Newman
[Full Article -
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3429-3429
| Fifty Years of Free Radicals By Cheves Walling. In Profiles, Pathways, and Dreams. Series Editor Jeffrey I. Seeman. American Chemical Society, Washington, D.C. 1995. xxiv + 141 pp. 15.5 × 23.5 cm. ISBN 0-8412-1830-7. $24.95.
Staff
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3429-3429
| Progress in Obesity Research: 7 Edited by A. Angel, H. Anderson, C. Bouchard, D. Lau, L. Leiter, and R. Mendelson. John Libbey & Co., Ltd., London. 1996. xvi + 768 pp. 17.5 × 24.5 cm. ISBN 0-86196-532-9.  70.00.
Staff
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3429-3430
| The chemistry of organophosphorus compounds. Volume 4. Ter- and quinque-valent phosphorus acids and their derivatives Edited by Frank P. Hartley. An Interscience Publication, John Wiley & Sons, Ltd., West Sussex, England. 1996. xiv + 945 pp. 16 × 24 cm. ISBN 0-471-95706-2. $375.00.
Staff
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3430-3430
| Adrenoceptors, Structure, Function and Pharmacology Edited by Robert R. Ruffolo, Jr. Harwood Academic Publisher GmbH, Distributed by University of Toronto Press, Toronto, Canada. 1995. xi + 279 pp. 18 × 25.5 cm. ISBN 3-7186-5644-2. $95.00.
Pieter B. M. W. M. Timmermans
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3430-3430
| Books of Interest
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