Journal of Medicinal Chemistry
Volume 39, Issue 24 (November 22, 1996)
Copyright © 1996
American Chemical Society
4689-4691 | Sustained Decrease in Cocaine-Maintained Responding in Rhesus Monkeys with 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]- 4-(3-hydroxy-3-phenylpropyl)piperazinyl Decanoate, a Long-Acting Ester Derivative of GBR 12909
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4692-4703 | Synthesis and Evaluation of Heterocyclic Carboxamides as Potential Antipsychotic Agents
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4704-4716 | Development of Novel, Potent, and Selective Dopamine Reuptake Inhibitors through Alteration of the Piperazine Ring of 1-[2-(Diphenylmethoxy)ethyl]- and 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazines (GBR 12935 and GBR 12909)
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4717-4726 | 5-HT1D Receptor Agonist Properties of Novel 2-[5-[[(Trifluoromethyl)sulfonyl]oxy]indolyl]ethylamines and Their Use as Synthetic Intermediates
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4727-4737 | Understanding the Binding of 5-Substituted 2'-Deoxyuridine Substrates to Thymidine Kinase of Herpes Simplex Virus Type-1
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4738-4743 | Diastereoselective Synthesis of All Four Isomers of 3-(4-Chlorophenyl)glutamic Acid: Identification of the Isomers Responsible for the Potentiation of L-Homocysteic Acid-Evoked Depolarizations in Neonatal Rat Motoneurons
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4744-4749 | Synthesis and Dopamine Transporter Affinity of 2-(Methoxycarbonyl)-9-methyl-3-phenyl-9-azabicyclo[3.3.1]nonane Derivatives
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4750-4755 | Computation of Brain-Blood Partitioning of Organic Solutes via Free Energy Calculations
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4756-4761 | Synthesis and Selective Monoamine Oxidase B-Inhibiting Properties of 1-Methyl-1,2,3,6-tetrahydropyrid-4-yl Carbamate Derivatives: Potential Prodrugs of (R)- and (S)-Nordeprenyl
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4762-4766 | Synthesis and Cytotoxic and Antitumor Activity of Esters in the 1,2-Dihydroxy-1,2-dihydroacronycine Series
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4767-4774 | Structure-Activity Relationship Studies on Benzofuran Analogs of Propafenone-Type Modulators of Tumor Cell Multidrug Resistance
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4775-4782 | Brain-Targeted Delivery of a Leucine-enkephalin Analogue by Retrometabolic Design
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4783-4803 | Glucose Transport-Enhancing and Hypoglycemic Activity of 2-Methyl-2-phenoxy-3-phenylpropanoic Acids
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4804-4809 | [125I/127I]IodoHoechst 33342: Synthesis, DNA Binding, and Biodistribution
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4810-4824 | Molecular Dynamics Simulations of the Bis-Intercalated Complexes of Ditercalinium and Flexi-Di with the Hexanucleotide d(GCGCGC)2: Theoretical Analysis of the Interaction and Rationale for the Sequence Binding Specificity
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4825-4832 | Solution of the Conformation and Alignment Tensors for the Binding of Trimethoprim and Its Analogs to Dihydrofolate Reductase: 3D-Quantitative Structure-Activity Relationship Study Using Molecular Shape Analysis, 3-Way Partial Least-Squares Regression, and 3-Way Factor Analysis
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4833-4843 | 1-Aminocyclobutanecarboxylic Acid Derivatives as Novel Structural Elements in Bioactive Peptides: Application to Tuftsin Analogs
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4844-4852 | Synthesis and Biological Activity of Conformationally Restricted Analogs of Milnacipran: (1S,2R)-1-Phenyl-2-[(S)-1-aminopropyl]-N,N-diethylcyclopropanecarboxamide, an Efficient Noncompetitive N-Methyl-D-aspartic Acid Receptor Antagonist
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4853-4859 | Estrogenic Triarylethylene Acetic Acids: Effect of Structural Variation on Estrogen Receptor Affinity and Estrogenic Potency and Efficacy in MCF-7 Cells
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4860-4866 | Nudicauline and Elatine as Potent Norditerpenoid Ligands at Rat Neuronal  -Bungarotoxin Binding Sites: Importance of the 2-(Methylsuccinimido)benzoyl Moiety for Neuronal Nicotinic Acetylcholine Receptor Binding
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