2793-2809
| New Approaches to Antiglaucoma Therapy
Michael F. Sugrue
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2810-2812
| 12,13-Isotaxanes: Synthesis of New Potent Analogs and X-ray Crystallographic Confirmation of Structure
Roy A. Johnson,
Paul J. Dobrowolski,
Eldon G. Nidy,
Ilse Gebhard,
Samuel J. Qualls,
Nancy A. Wicnienski,
Robert C. Kelly,
Thomas W. Pitts,
Narima M. Lopes,
Thomas F. DeKoning,
Sally J. Mattern,
Sheldon D. Weed,
J. Patrick McGovren, and
Constance G. Chidester
[Full Article -
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2813-2817
| Selective Inhibition of Neuronal Nitric Oxide Synthase by N -Nitroarginine- and Phenylalanine-Containing Dipeptides and Dipeptide Esters
Richard B. Silverman,
Hui Huang,
Michael A. Marletta, and
Pavel Martasek
[Full Article -
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2818-2824
| Terbenzimidazoles: Influence of 2''-, 4-, and 5-Substituents on Cytotoxicity and Relative Potency as Topoisomerase I Poisons
Jung Sun Kim,
Chiang Yu,
Angela Liu,
Leroy F. Liu, and
Edmond J. LaVoie
[Full Article -
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2825-2830
| Synthesis of Carboranes Containing an Azulene Framework and in Vitro Evaluation as Boron Carriers
Hiroyuki Nakamura,
Masaru Sekido, and
Yoshinori Yamamoto
[Full Article -
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2831-2842
| Heteroaryl Analogues of AMPA. Synthesis and Quantitative Structure-Activity Relationships
Benny Bang-Andersen,
Sibylle M. Lenz,
Niels Skjærbæk,
Karina K. S by,
Hans O. Hansen,
Bjarke Ebert,
Klaus P. Bges, and
Povl Krogsgaard-Larsen
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2843-2857
| Use of Conformationally Restricted Benzamidines as Arginine Surrogates in the Design of Platelet GPIIb-IIIa Receptor Antagonists
Daniel J. Sall,
Ann E. Arfsten,
Jolie A. Bastian,
Michael L. Denney,
Cathy S. Harms,
Jefferson R. McCowan,
John M. Morin, Jr.,
Jack W. Rose,
Robert M. Scarborough,
Mark S. Smyth,
Suzane L. Um,
Barbara G. Utterback,
Robert T. Vasileff,
James H. Wikel,
Virginia L. Wyss, and
Joseph A. Jakubowski
[Full Article -
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2858-2865
| Novel Biological Response Modifiers: Phthalimides with Tumor Necrosis Factor- Production-Regulating Activity
Hiroyuki Miyachi,
Akihiko Azuma,
Asuka Ogasawara,
Eiji Uchimura,
Naoko Watanabe,
Yoshiro Kobayashi,
Fuminori Kato,
Masanari Kato, and
Yuichi Hashimoto
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2866-2875
| Substituted (Pyridylmethoxy)naphthalenes as Potent and Orally Active 5-Lipoxygenase Inhibitors: Synthesis, Biological Profile, and Pharmacokinetics of L-739,010
Pierre Hamel,
Denis Riendeau,
Christine Brideau,
Chi-Chung Chan,
Sylvie Desmarais,
Daniel Delorme,
Daniel Dubé,
Yves Ducharme,
Diane Ethier,
Erich Grimm,
Jean-Pierre Falgueyret,
Jocelyne Guay,
Tom R. Jones,
Elizabeth Kwong,
Malia McAuliffe,
Cyril S. McFarlane,
Hanna Piechuta,
Marie Roumi,
Philip Tagari,
Robert N. Young, and
Yves Girard
[Full Article -
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2876-2882
| Design of Low Molecular Weight Hematoregulatory Agents from the Structure-Activity Relationship of a Dimeric Pentapeptide
Alan S. Cuthbertson,
Mette Husbyn,
May Engebretsen,
Michael Hartmann,
Meinolf Lange,
Jessie Sandosham,
Peter M. Fischer,
Hege Fjerdingstad, and
Dagfinn Lvhaug
[Full Article -
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2883-2894
| Synthesis and Activity of 6-Substituted Purine Linker Amino Acid Immunostimulants
Boulos Zacharie,
Lyne Gagnon,
Giorgio Attardo,
Timothy P. Connolly,
Yves St-Denis, and
Christopher L. Penney
[Full Article -
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2895-2901
| Total Syntheses and Anticholinesterase Activities of (3aS)-N(8)-Norphysostigmine, (3aS)-N(8)-Norphenserine, Their Antipodal Isomers, and Other N(8)-Substituted Analogues
Qian-sheng Yu,
Xue-Feng Pei,
Harold W. Holloway, and
Nigel H. Greig
, Arnold Brossi
[Full Article -
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2902-2909
| O6-(Alkyl/aralkyl)guanosine and 2'-Deoxyguanosine Derivatives: Synthesis and Ability To Enhance Chloroethylnitrosourea Antitumor Action
Emmanuelle Mounetou,
Eric Debiton,
Catherine Buchdahl,
Daniel Gardette,
Jean-Claude Gramain,
Jean-Claude Maurizis,
Annie Veyre, and
Jean-Claude Madelmont
[Full Article -
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2910-2921
| Mapping the Peripheral Benzodiazepine Receptor Binding Site by Conformationally Restrained Derivatives of 1-(2-Chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide (PK11195)
Andrea Cappelli,
Maurizio Anzini,
Salvatore Vomero,
Pier G. De Benedetti,
Maria Cristina Menziani,
Gianluca Giorgi, and
Cristina Manzoni
[Full Article -
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2922-2930
| Synthesis and Structure-Activity Relationships of 6,7-Benzomorphan Derivatives as Antagonists of the NMDA Receptor-Channel Complex
Matthias Grauert,
Wolf Dietrich Bechtel,
Helmut A. Ensinger,
Herbert Merz, and
Adrian J. Carter
[Full Article -
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2931-2935
| (S)-Spiro[(1,3-diazacyclopent-1-ene)-5,2'-(7'-methyl-1',2',3',4'- tetrahydronaphthalene)]: Resolution, Stereospecific Synthesis, and Preliminary Pharmacological Characterization as a Partial -Adrenergic Agonist
Alex A. Cordi,
Jean-Michel Lacoste,
Fabrice Le Borgne,
Yolande Herve,
Lucile Vaysse-Ludot,
Jean-Jacques Descombes,
Christine Courchay,
Michel Laubie, and
Tony J. Verbeuren
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2936-2947
| Probes for Narcotic Receptor-Mediated Phenomena. 25. Synthesis and Evaluation of N-Alkyl-Substituted (-Piperazinylbenzyl)benzamides as Novel, Highly Selective  Opioid Receptor Agonists
Yousuke Katsura,
Xiaoyan Zhang,
Koichi Homma,
Kenner C. Rice,
Silvia N. Calderon,
Richard B. Rothman,
Henry I. Yamamura,
Peg Davis,
Judith L. Flippen-Anderson,
Heng Xu,
Karen Becketts,
Eric J. Foltz, and
Frank Porreca
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2948-2952
| Synthesis and Pharmacological Activity of Deltorphin and Dermorphin-Related Glycopeptides
Roberto Tomatis,
Mauro Marastoni,
Gianfranco Balboni,
Remo Guerrini,
Anna Capasso,
Ludovico Sorrentino,
Vincenzo Santagada,
Giuseppe Caliendo,
Lawrence H. Lazarus, and
Severo Salvadori
[Full Article -
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2953-2958
| A Theoretical Investigation of Tight-Binding Thermolysin Inhibitors
Jian Shen
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2959-2966
| Synthesis and Properties of Second-Generation 2-5A-Antisense Chimeras with Enhanced Resistance to Exonucleases
Guiying Li,
Wei Xiao, and
Paul F. Torrence
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2967-2967
| Biomedical Frontiers of Fluorine Chemistry Edited by Iwao Ojima, James R. McCarthy, and John T. Welch. ACS Symposium Series No. 639. 1996. xi + 356 pp. 15.5 × 23.5 cm. ISBN 0-8412-3442-6. $99.95.
Adeboye Adejare
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2967-2968
| Genetic Algorithms in Molecular Modeling Edited by J. Devillers. Academic Press, London. 1996. x + 327 pp. 15.5 × 23.5 cm. ISBN 0-12-213810-4. $55.00.
Lemont B. Kier
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2968-2968
| Biological NMR Spectroscopy Edited by John L. Markley and Stanley J. Opella. Oxford University Press, New York, 1997. x + 360 pp. 16 × 24 cm. ISBN 0-19-509468-9. $65.00.
Rickey P. Hicks
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2968-2969
| Encyclopedia of Cancer. Volumes 1-3 Edited by Joseph R. Bertino. Academic Press, Inc., San Diego, CA. 1997. xxxviii + 2134 pp. 22.5 × 28.5 cm. ISBN 0-12-093-230-X. $475.00 (3 volume set).
Janice R. Sufrin
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2969-2969
| Molecular Modeling: Principles and Applications By Andrew Leach. Longman, Edinburgh. 1996. xvi + 595 pp. ISBN 0-582-23933-8. $35.00.
Lemont B. Kier
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2969-2970
| Neural Networks in QSAR and Drug Design Edited by J. Devillers. Academic Press, London. 1996. x + 284 pp. 15.5 × 23.5 cm. ISBN 0-12-213815-5. $65.00.
Lemont B. Kier
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2970-2970
| The Ionotropic Glutamate Receptors Edited by Daniel T. Monaghan and Robert J. Wenthold. Humana Press, Totowa, NJ. 1997. x + 378 pp. 16 × 23.5 cm. ISBN 0-89603-4756-9. $135.00.
John Wm. Ferkany
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