Journal of Medicinal Chemistry
Volume 41, Issue 3 (January 29, 1998)
Copyright © 1998
American Chemical Society
| COMMUNICATIONS TO THE EDITOR | |
263-265 | Novel Potent Nonpeptide Aminopeptidase N Inhibitors with a Cyclic Imide Skeleton
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266-270 | Striking Effect of Hydroxamic Acid Substitution on the Phosphodiesterase Type 4 (PDE4) and TNF Inhibitory Activity of Two Series of Rolipram Analogues: Implications for a New Active Site Model of PDE4
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271-275 | Binding of ATP-Sensitive Potassium Channel (KATP) Openers to Cardiac Membranes: Correlation of Binding Affinities with Cardioprotective and Smooth Muscle Relaxing Potencies
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ARTICLES | |
276-283 | Synthesis and Biodistribution of a Short Nonionic Oligonucleotide Analogue in Mouse with a Potential to Mimic Peptides
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284-290 | Design of N-Acylprolyltyrosine "Tripeptoid" Analogues of Neurotensin as Potential Atypical Antipsychotic Agents
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291-302 | 5-Aryl-1,2-dihydrochromeno[3,4-f]quinolines: A Novel Class of Nonsteroidal Human Progesterone Receptor Agonists
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303-310 | 5-Aryl-1,2-dihydro-5H-chromeno[3,4-f]quinolines as Potent, Orally Active, Nonsteroidal Progesterone Receptor Agonists: The Effect of D-Ring Substituents
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311-317 | 5-HT3 Antagonists Derived from Aminopyridazine-type Muscarinic M1 Agonists
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318-331 | Synthesis, Pharmacological Characterization, and Quantitative Structure-Activity Relationship Analyses of 3,7,9,9-Tetraalkylbispidines: Derivatives with Specific Bradycardic Activity
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332-338 | cis-[PtCl2(4,7-H-5-methyl-7-oxo[1,2,4]triazolo[1,5-a]pyrimidine)2]: A Sterically Restrictive New Cisplatin Analogue. Reaction Kinetics with Model Nucleobases, DNA Interaction Studies, Antitumor Activity, and Structure-Activity Relationships
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339-345 | Design and Synthesis of Malonic Acid-Based Inhibitors of Human Neutrophil Collagenase (MMP8)
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346-357 | 2-Substituted (2SR)-2-Amino-2-((1SR,2SR)-2-carboxycycloprop-1-yl)glycines as Potent and Selective Antagonists of Group II Metabotropic Glutamate Receptors. 1. Effects of Alkyl, Arylalkyl, and Diarylalkyl Substitution
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358-378 | 2-Substituted (2SR)-2-Amino-2-((1SR,2SR)-2-carboxycycloprop-1-yl)glycines as Potent and Selective Antagonists of Group II Metabotropic Glutamate Receptors. 2. Effects of Aromatic Substitution, Pharmacological Characterization, and Bioavailability
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379-392 | 1,2,5-Thiadiazole Analogues of Aceclidine as Potent m1 Muscarinic Agonists
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393-400 | Quantitative Analysis of the Structural Requirements for Blockade of the N-Methyl-D-aspartate Receptor at the Phencyclidine Binding Site
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NOTES | |
401-406 | Discovery and Development of the Novel Potent Orally Active Thrombin Inhibitor N-(9-Hydroxy-9-fluorenecarboxy)prolyl trans-4-Aminocyclohexylmethyl Amide (L-372,460): Coapplication of Structure-Based Design and Rapid Multiple Analogue Synthesis on Solid Support
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