Journal of Medicinal Chemistry
Volume 42, Issue 6 (March 25, 1999)
Copyright © 1999
American Chemical Society
| COMMUNICATIONS TO THE EDITOR | |
947-950 | Postsynthetic Generation of a Major Acrolein Adduct of 2'-Deoxyguanosine in Oligomeric DNA
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EXPEDITED ARTICLES | |
951-956 | Novel Inhibitors of Carboxypeptidase G2 (CPG2): Potential Use in Antibody-Directed Enzyme Prodrug Therapy
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ARTICLES | |
957-962 | Design, Synthesis, and Evaluation of Conformationally Constrained Tongs, New Inhibitors of HIV-1 Protease Dimerization
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963-970 | Structure-Activity Relationships of Lysophosphatidic Acid: Conformationally Restricted Backbone Mimetics
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971-980 | Structural and Conformational Requirements for High-Affinity Binding to the SH2 Domain of Grb2
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981-991 | 6-Substituted Benzopyrans as Potassium Channel Activators: Synthesis, Vasodilator Properties, and Multivariate Analysis
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992-998 | Diversity Analysis of 14 156 Molecules Tested by the National Cancer Institute for Anti-HIV Activity Using the Quantitative Structure-Activity Relational Expert System MCASE
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999-1006 | Cytotoxicity of (2,2':6',2' '-Terpyridine)platinum(II) Complexes to Leishmania donovani, Trypanosoma cruzi, and Trypanosoma brucei
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1007-1017 | Synthesis and Antiparasitic and Antitumor Activity of 2,4-Diamino-6-(arylmethyl)-5,6,7,8-tetrahydroquinazoline Analogues of Piritrexim
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1018-1026 | Use of a Pharmacophore Model for the Design of EGFR Tyrosine Kinase Inhibitors: Isoflavones and 3-Phenyl-4(1H)-quinolones
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1027-1040 | Synthesis, Pharmacological Characterization, and Molecular Modeling of Heterobicyclic Amino Acids Related to (+)-2-Aminobicyclo[3.1.0]hexane- 2,6-dicarboxylic Acid (LY354740): Identification of Two New Potent, Selective, and Systemically Active Agonists for Group II Metabotropic Glutamate Receptors
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1041-1052 | Structure-Activity Relationship of Diaryl Phosphonate Esters as Potent Irreversible Dipeptidyl Peptidase IV Inhibitors
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1053-1065 | Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)
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1066-1075 | Glutathione-Mediated Metabolism of Technetium-99m SNS/S Mixed Ligand Complexes: A Proposed Mechanism of Brain Retention
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1076-1087 | Design, Synthesis, Structure-Activity Relationships, and Biological Characterization of Novel Arylalkoxyphenylalkylamine  Ligands as Potential Antipsychotic Drugs
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1088-1099 | Novel, Potent, and Selective Phosphodiesterase-4 Inhibitors as Antiasthmatic Agents: Synthesis and Biological Activities of a Series of 1-Pyridylnaphthalene Derivatives
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BRIEF ARTICLES | |
1100-1105 | Melatonergic Properties of the (+)- and (-)-Enantiomers of N-(4-Methoxy-2,3-dihydro-1H-phenalen-2-yl)amide Derivatives
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1106-1111 | Thieno[3,2-b]- and Thieno[2,3-b]pyrrole Bioisosteric Analogues of the Hallucinogen and Serotonin Agonist N,N-Dimethyltryptamine
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BOOK REVIEWS | |
1112-1112 | Metal-catalyzed Cross-coupling Reactions Edited by François Diederich and Peter J. Stang. Wiley-VCH, Weinheim. 1998. xxi + 517 pp. 17 × 25 cm. ISBN 3-527-29421-X. $140.00.
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1112-1113 | Structure-based Ligand Design Edited by K. Gubernator and H.-J. Bohm. Wiley-VCH, Weinheim. 1998. xiv + 153 pp. 17.5 × 24.5 cm. ISBN 3-527-29343-4. $135.00.
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1113-1113 | Strategies for Organic Drug Synthesis and Design By Daniel Lednicer. John Wiley & Sons, Inc., New York. 1998. xv + 502 pp. 16.5 × 24 cm. ISBN 0-471-19657-6. $79.95.
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ADDITIONS AND CORRECTIONS | |
1114-1114 | Bis- and Mixed-Tetrahydroisoquinolinium Chlorofumarates: New Ultra-Short-Acting Nondepolarizing Neuromuscular Blockers
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