EDITORIAL
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4927-4927
A Flexible Policy Concerning Purity Criteria for Published Target Compounds
Philip S. Portoghese
Editor-in-Chief
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COMMUNICATIONS
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4928-4931
Inhibitors of Efflux Pumps in Pseudomonas aeruginosa Potentiate the Activity of the Fluoroquinolone Antibacterial Levofloxacin
Thomas E. Renau,
Roger Léger,
Eric M. Flamme,
Joan Sangalang,
Miles W. She,
Rose Yen,
Carla L. Gannon,
David Griffith,
Suzanne Chamberland,
Olga Lomovskaya,
Scott J. Hecker,
Ving J. Lee,
Toshiharu Ohta, and
Kiyoshi Nakayama
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ARTICLES
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4932-4941
Structure-Activity Studies of Cerulenin Analogues as Protein Palmitoylation Inhibitors
David S. Lawrence,
Jack T. Zilfou, and
Charles D. Smith
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4942-4951
Designing Libraries with CNS Activity
Ajay,
Guy W. Bemis, and
Mark A. Murcko
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4952-4960
On the Bioactive Conformation of NAN-190 (1) and MP3022 (2), 5-HT1A Receptor Antagonists
Maria H. Paluchowska,
Maria J. Mokrosz,
Andrzej Bojarski,
Anna Wesoowska,
Jolanta Borycz,
Sijka Charakchieva-Minol, and
Ewa Chojnacka-Wójcik
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4961-4969
Structure-Activity Relationship Studies of Novel Heteroretinoids: Induction of Apoptosis in the HL-60 Cell Line by a Novel Isoxazole-Containing Heteroretinoid
Daniele Simoni,
Francesco Paolo Invidiata,
Riccardo Rondanin,
Stefania Grimaudo,
Giuliana Cannizzo,
Eleonora Barbusca,
Ferdinando Porretto,
Nicola D'Alessandro, and
Manlio Tolomeo
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4970-4980
Improving the Nicotinic Pharmacophore with a Series of (Isoxazole)methylene-1-azacyclic Compounds: Synthesis, Structure-Activity Relationship, and Molecular Modeling
Janne E. Tnder,
John Bondo Hansen,
Mikael Begtrup,
Ingrid Pettersson,
Karin Rimvall,
Birgitte Christensen,
Ulrich Ehrbar, and
Preben H. Olesen
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4981-5001
3-[3-(Piperidin-1-yl)propyl]indoles as Highly Selective h5-HT1D Receptor Agonists
Michael G. N. Russell,
Victor G. Matassa,
Roy R. Pengilley,
Monique B. van Niel,
Bindi Sohal,
Alan P. Watt,
Laure Hitzel,
Margaret S. Beer,
Josephine A. Stanton,
Howard B. Broughton, and
José L. Castro
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5002-5009
Chemical Syntheses and Biological Studies on Dimeric Chimeras of Oxytocin and the V2-Antagonist, d(CH2)5[D-Ile2,Ile4]arginine Vasopressin
Lin Chen,
Regina Golser,
Alena Machová,
Jirina Slaninová, and
George Barany
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5010-5019
Further Studies on the Dmt-Tic Pharmacophore: Hydrophobic Substituents at the C-Terminus Endow Antagonists To Manifest Agonism or Antagonism
Severo Salvadori,
Remo Guerrini,
Gianfranco Balboni,
Clementina Bianchi,
Sharon D. Bryant,
Peter S. Cooper, and
Lawrence H. Lazarus
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5020-5028
Benzimidazole Derivatives. 2. Synthesis and Structure-Activity Relationships of New Azabicyclic Benzimidazole-4-carboxylic Acid Derivatives with Affinity for Serotoninergic 5-HT3 Receptors
María L. López-Rodríguez,
Bellinda Benhamú,
M. José Morcillo,
Ignacio D. Tejada,
Luis Orensanz,
M. José Alfaro, and
M. Isabel Martín
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5029-5042
Oxygenated Analogues of 1-[2-(Diphenylmethoxy)ethyl]- and 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazines (GBR 12935 and GBR 12909) as Potential Extended-Action Cocaine-Abuse Therapeutic Agents
David B. Lewis,
Dorota Matecka,
Ying Zhang,
Ling-Wei Hsin,
Christina M. Dersch,
David Stafford,
John R. Glowa,
Richard B. Rothman, and
Kenner C. Rice
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5043-5052
Synthesis and in Vitro Evaluation of New 8-Amino-1,4-benzoxazine Derivatives as Neuroprotective Antioxidants
Martine Largeron,
Brian Lockhart,
Bruno Pfeiffer, and
Maurice-Bernard Fleury
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5059-5059
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5053-5058
Bisphosphonate Prodrugs: Synthesis and in Vitro Evaluation of Novel Acyloxyalkyl Esters of Clodronic Acid
Riku Niemi,
Jouko Vepsäläinen,
Hannu Taipale, and
Tomi Järvinen
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BOOK REVIEWS
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ADDITIONS AND CORRECTIONS
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5060-5060
High-Resolution NMR and Computer Modeling Studies of the Cannabimimetic Aminoalkylindole Prototype WIN-55212-2
Xiang-Qun Xie,
Xiu-Wen Han,
Jian-Zhong Chen,
Michael Eissenstat, and
Alexandros Makriyannis
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