641-659
Perspectives in Animal Health: Old Targets and New Opportunities
660-663
X-ray Structure of Citrate Bound to Src SH2 Leads to a High-Affinity, Bone-Targeted Src SH2 Inhibitor
ARTICLES
664-671
Anti-AIDS Agents. 42. Synthesis and Anti-HIV Activity of Disubstituted (3'R,4'R)-3',4'-Di-O-(S)-camphanoyl-(+)-cis-khellactone Analogues
672-680
A New Class of Nonsteroidal Aromatase Inhibitors: Design and Synthesis of Chromone and Xanthone Derivatives and Inhibition of the P450 Enzymes Aromatase and 17 
-Hydroxylase/C17,20-Lyase
681-693
Discovery of 4-[3-(trans-3-Dimethylaminocyclobutyl)-1H-indol-5-ylmethyl]- (4S)-oxazolidin-2-one (4991W93), a 5HT1B/1D Receptor Partial Agonist and a Potent Inhibitor of Electrically Induced Plasma Extravasation
694-702
Antimitotic Antitumor Agents: Synthesis, Structure-Activity Relationships, and Biological Characterization of N-Aryl-N'-(2-chloroethyl)ureas as New Selective Alkylating Agents
703-714
Correlation of Anti-HIV Activity with Anion Spacing in a Series of Cosalane Analogues with Extended Polycarboxylate Pharmacophores
715-724
Heterobifunctional Ligands: Practical Chemoenzymatic Synthesis of a Cell Adhesive Glycopeptide That Interacts with Both Selectins and Integrins
725-736
Cyclic Ketone Inhibitors of the Cysteine Protease Cathepsin K
737-748
Design, Synthesis, and Evaluation of a Novel Pyrrolobenzodiazepine DNA-Interactive Agent with Highly Efficient Cross-Linking Ability and Potent Cytotoxicity
749-762
Thiazole and Thiadiazole Analogues as a Novel Class of Adenosine Receptor Antagonists
763-768
C-Isoprenylation of Flavonoids Enhances Binding Affinity toward P-Glycoprotein and Modulation of Cancer Cell Chemoresistance
769-776
Electrooxidation Potential as a Tool in the Early Screening for New Safer Clozapine-like Analogues
777-786
New 3'-Azido-3'-deoxythymidin-5'-yl O-( 
-Hydroxyalkyl) Carbonate Prodrugs: Synthesis and Anti-HIV Evaluation
787-805
Potential Antidepressants Displayed Combined 2-Adrenoceptor Antagonist and Monoamine Uptake Inhibitor Properties
806-813
Syntheses and Structure-Activity Relationships of Novel Apio and Thioapio Dideoxydidehydronucleosides as Anti-HCMV Agents
814-821
Antipsoriatic Anthrones with Modulated Redox Properties. 5. Potent Inhibition of Human Keratinocyte Growth, Induction of Keratinocyte Differentiation, and Reduced Membrane Damage by Novel 10-Arylacetyl-1,8-dihydroxy-9(10H)-anthracenones
822-833
Synthesis and Src Kinase Inhibitory Activity of a Series of 4-Phenylamino-3-quinolinecarbonitriles
834-848
Syntheses and Biological Activities of a Novel Group of Steroidal Derived Inhibitors for Human CDC25A Protein Phosphatase
BOOK REVIEWS
849-849
CRC Handbook of Laboratory Safety. 5th Edition By A. Keith Furr. CRC Press, Boca Raton, FL. 2000. xvii + 774 pp. 18 × 26 cm. ISBN 0-8493-2523-4. $149.99.
849-850
Methods in Molecular Biology, Volume 146. Mass Spectrometry of Proteins and Peptides Edited by John R. Chapman. Humana Press, Totowa, NJ. 2000. xiv + 538 pp. 15.5 × 23.5 cm. ISBN 0-89603-609-x. $125.00.
850-850
Biodiversity. New Leads for the Pharmaceutical and Agrochemical Industries Edited by Stephen K. Wrigley, Martin A. Hayes, Robert Thomas, Ewan J. T. Chrystal, and Neville Nicholson. The Royal Society of Chemistry, Cambridge, U.K. 2000. vi + 314 pp. 16 × 24 cm. ISBN 0-85404-830-8. 
59.50.