Journal of Heterocyclic Chemistry Table of Contents: 2012, vol. 49, No. 4

Highlight: Stereoselective Cross-Dehydrogenative Coupling Reactions Based on Sp3 C―H Activation to Give Chiral Heterocyclic Compounds
Ming Zhang and Aiqin Zhang
721-725

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An Efficient Synthesis of Thiazolidine-4-ones with Antitumor and Antioxidant Activities
Ashraf A. Aly, Alan B. Brown, Mohamed Abdel-Aziz, Gamal El-Din A. A. Abuo-Rahma, Mohamed F. Radwan, Mohamed Ramadan and Amira M. Gamal-Eldeen
726-731

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Synthesis and Herbicidal Activity of Acylpyrazole Derivatives Containing 1,2,3-Thiadiazole Moiety
Feng Cheng and De-Qing Shi
732-736

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Synthesis and Functionalization of 8-Methyl-2h-pyrimido [2,1-c][1,2,4]triazine-3,6(1h,4h)-dione
Virginija Jakubkiene, Vytautas Cepla, Milda M. Burbuliene and Povilas Vainilavicius
737-741

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Polycyclic N-Heterocyclic Compounds, Part 71: Synthesis and Bronchodilator Evaluation of 5-Substituted 1,2-Dihydrofuro[3,2-f][1,7]naphthyridines and Related Compounds
Kensuke Okuda, Tetsuo Matsushita, Takashi Hirota and Kenji Sasaki
742-747

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Synthesis of Some Novel Pyrazole-Substituted 9-Anilinoacridine Derivatives and Evaluation for their Antioxidant and Cytotoxic Activities
R. Kalirajan, V. Muralidharan, S. Jubie, B. Gowramma, S. Gomathy, S. Sankar and K. Elango
748-754

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Polycyclic N-Heterocyclic Compounds, Part 72: Reaction of N-([1]Benzofuro (or Benzothieno)[3,2-d]pyrimidin-4-yl)formamidine and N-(Pyrido[2,3-d]pyrimidin-4-yl)formamidine Derivatives with Hydroxylamine Hydrochloride
Kensuke Okuda, Kiyoko Tsuchie and Takashi Hirota
755-762

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Synthesis and Structure of 3,4-Dihydropyrido[2′,3′:3,4]pyrazolo[1,5-a][1,3,5]triazin-2-amines
Anton V. Dolzhenko, Shiqi Bai, Anna V. Dolzhenko and Wai Keung Chui
763-767

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General Two-Step Preparation of Chalcones Containing Thiazole
Dagobert Tazoo, Ovidiu Oniga, D. Scott Bohle, Zhijie Chua and Etienne Dongo
768-773

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Utility of Enaminonitriles in Heterocyclic Synthesis: Synthesis of Some New Pyrazole, Pyridine, and Pyrimidine Derivatives
Ahmed A. Fadda, Hassan A. Etman, Mohamed Y. El-Seidy and Khaled M. Elattar
774-781

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A Theoretical Study of NBO, NICS, and 14N NQR Parameters of Adenine Tautomers in the Gas Phase via DFT
Ehsan Zahedi
782-788

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A Facile One-Pot Synthesis of Substituted Quinolines via New Multicomponent Reaction
Amir Rineh, Mohammad A. Khalilzadeh, Mohammad M. Hashemi, Medí Rajabi and Fatemeh Karimi
789-791

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Synthesis and Antiproliferative Evaluation of 2′-Arenesulfonyloxy-5-benzylidene-thiazolidine-2,4-diones
Emily M. Chen, Pei-Jung Lu and Arthur Y. Shaw
792-798

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Synthesis of New PMB-Substituted Indoles Containing 1,3,4-Oxadiazole and 1,2,4-Triazole Units
Abdel-Rahman Farghaly, Norbert Haider and Duck-Hyung Lee
799-805

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Benzimidazole Annulated New Heterocyclic Compounds: Synthesis of New Polycyclic Pyrazole Derivatives
Mohamed Ali A. Khalil
806-813

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Synthesis and NMR Spectroscopic Characteristics of a Series of Hydrazide-Hydrazones Containing Furoxan Ring Derived from Isoeugenoxyacetic Acid
Nguyen Huu Dinh, Hoang Thi Tuyet Lan, Tran Thi Thu Trang and Pham Van Hoan
814-822

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Facile Synthesis of 3,6-Disubstituted-1,2,4-triazolo-[3,4-b]-1,3,4-thiadiazoles via Oxidative Cyclization of n-Heteroaryl-Substituted Hydrazones and Their Biological Activity
M. Himaja, K. Jagadeesh Prathap and Sunil V. Mali
823-828

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CNS-Agent Precursor: A Simple and Efficient Synthesis of an Antipsychotic Drug Fluanisone
A. Venkat Narsaiah, B. Nagaiah and B. Karuna Devi
829-832

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(Bromodimethyl)sulfonium Bromide Catalyzed Solvent-Free Friedlander Synthesis of Substituted Quinolines
R. Venkatesham, A. Manjula and B. Vittal Rao
833-838

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Syntheses, Characterization, and Antibacterial Activities of Four New Schiff Base Compounds Derived from 1-Phenyl-3-methyl-4-benzoyl-2-pyrazolin-5-one
Chong-Bo Liu, Yuan Chen, Liu-Shui Yan, De-He Huang and Zhi-Qiang Xiong
839-844

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The Synthesis of 3-Amino-pyrazine-2-carbohydrazide and 3-Amino-N′-methylpyrazine-2-carbohydrazide Derivatives
Barbara Milczarska, Katarzyna Gobis, Henryk Foks, Lukasz Golunski and Pawel Sowinski
845-850

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Practical and Green Protocol for the Synthesis of Substituted 4H-Chromenes Using Room Temperature Ionic Liquid Choline Chloride–Urea
C. N. Revanna, T. R. Swaroop, G. M. Raghavendra, D. G. Bhadregowda, K. Mantelingu and K. S. Rangappa
851-855

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Synthesis of Novel 5,6-Dihydropyrrolo[2,1-a]isoquinolines via Grob Reaction between (E)-1,1,1-Trifluoro-3-nitro-2-butene and 3,4-Dihydroisoquinolines
Vladislav Y. Korotaev, Vyacheslav Y. Sosnovskikh, Alexey Y. Barkov, Pavel A. Slepukhin and Yurii V. Shklyaev
856-860

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Methanesulfonic Acid-Catalyzed One-Pot Synthesis of 12-Aryl or 12-Alkyl-8,9,10,12-tetrahydrobenzo[a]xanthen-11-one Derivatives
Yu-Heng Liu and Lei Li
861-864

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Synthesis of N-Substituted-6-alkoxypteridin-4-amine
Chonggang Duan, Jiong Jia, Rongxiu Zhu and Jianwu Wang
865-872

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Novel Synthesis and Antimicrobial Activity of 3-Substituted 5-bromo-7-methyl-1,2,4-triazolo-[3,4-b]-benzothiazoles
T. M. Bhagat, S. K. Deshmukh and S. V. Kuberkar
873-876

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Microwave-Assisted Solvent-Free Synthesis of Highly Functionalized Pyrimidine Derivatives
Shengjiao Yan, Yanfei Niu, Xuebing Chen, Yongjiang Liu and Jun Lin
877-882

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Isomeric 3-Isoxadiazolylcoumarins and Their Derivatives
Oleksandr S. Detistov, Valeriy D. Orlov and Irina O. Zhuravel'
883-892

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A Novel Synthesis of 4-Pyridazineacetic Acids via Ring Expansion of N-Cyanomethylated 3-Pyrazoline-4-acetic Acids
Eiichi Masumoto, Hiroshi Maruoka, Fumi Okabe, Sho Nishida, Ryoko Tomita, Toshihiro Fujioka and Kenji Yamagata
893-899

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Synthesis and Crystal Structure of 4,7-Diaryl-5-oxo-4H-benzo[b]pyran Derivatives
Bin Cui, Li-Zhuang Chen, Xiao-Lei Hu, Ming Wang and Guang-Fan Han
900-904

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Novel and Convenient Synthesis of Benzofurans from Dihydrocoumarins
Sharona Shachan-Tov and Aryeh A. Frimer
905-908

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Synthesis of Thieno[2,3-b]quinolinone Derivatives
Guang-Fan Han, Ming Wang, Li-Zhuang Chen and Xiao-Lei Hu
909-912

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An Improved Synthesis of Carbazoles via Domino Reaction of N-Protected-2-methylindoles with DMF-DMA/DMA-DMA
Radhakrishnan Sureshbabu and Arasambattu K. Mohanakrishnan
913-918

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A Re-Examination of the Reaction of 3,4-Diamino[1,2,5]oxadiazole with Glyoxal
Rodney L. Willer, Robson F. Storey, Christopher G. Campbell, Steven W. Bunte and Damon Parrish
919-925

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Preparation of Novel Di-isoxazolines Using Bis(nitrile oxide) 1,3-Dipolar Cycloaddition Methodology
Mohammad Ali Bigdeli, Azim Ziyaei Halimehjani, Mohammad Mohammadipour and Parishad Sagharichi
926-928

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Design, Synthesis, Characterization, and Antimicrobial Activity of Biginelli Products of Indandione
Vijay V. Dabholkar, Sunil R. Patil and Rajesh V. Pandey
929-932

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K2CO3/H2O in [omim][BF4] Ionic Liquid: A Green Medium for Efficient Room-Temperature Synthesis of N-Substituted 1,4-Benzoxazin-3-ones
Ali Sharifi, Mehdi Barazandeh, M. Saeed Abaee and Mojtaba Mirzaei
933-938

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Dithiocarbamates as an Efficient Intermediate for the Synthesis of Symmetrical Substituted 2,5-Diamino-1,3,4-thiadiazoles in Water
Azim Ziyaei Halimehjani, Akram Ashouri and Katayoun Marjani
939-942

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A Mild and Highly Efficient Synthesis of Chiral N-Dichloroacetyl-4-ethyl-1,3-oxazolidines
Li-Xia Zhao, Ying Fu, Fei Ye and Shuang Gao
943-946

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Conversion of Some 2(3H)-Furanones into Pyrrolinotriazine and Oxazolopyrimidine Derivatives
Wael S. I. Abou-Elmagd and Ahmed I. Hashem
947-950

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A Novel Method for the Synthesis of Spiro[indoline-Pyrazolo[4′,3′:5,6]pyrido[2,3-d]pyrimidine]triones by Alum as a Reusable Catalyst
Sadif A. Shirvan, Ramin Ghahremanzadeh, Mojtaba Mirhosseini Moghaddam, Ayoob Bazgir, Amir Hassan Zarnani and Mohammad Mehdi Akhondi
951-954

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Regioselective Synthesis of New Bibracchial Lariat Ethers
Sattar Ebrahimi, Akbar Mobinikhaldei and Naser Foroughifar
955-958

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A Novel and Efficient One Pot Synthesis of 2,4-Disubstituted Thiazoles and Oxazoles Using Phenyltrimethylammoniumtribromide in Ionic Liquid
Manoj Kumar Muthyala and Anil Kumar
959-964

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Acid Catalyzed tert-Butylation and Tritylation of 4-Nitro-1,2,3-triazole: Selective Synthesis of 1-Methyl-5-nitro-1,2,3-triazole via 1-tert-Butyl-4-nitro-1,2,3-triazole
Yuliya V. Filippova, Anna G. Sukhanova, Sergei V. Voitekhovich, Vadim E. Matulis, Gennady T. Sukhanov, Yury V. Grigoriev and Oleg A. Ivashkevich
965-968

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